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Signaling peptide receptor
Cell surface receptors
Cell surface receptors
Signaling peptide receptor is a type of receptor which binds one or more signaling peptides or signaling proteins.
An example is the tropomyosin receptor kinase B (TrkB), which is bound and activated by the neurotrophic protein brain-derived neurotrophic factor (BDNF). Another example is the μ-opioid receptor (MOR), which is bound and activated by the opioid peptide hormone β-endorphin.
Adiponectin receptor
Main article: Adiponectin receptor
AdipoR1
Main article: Adiponectin receptor 1
- Agonists
- Peptide
- Adiponectin
- ADP-355
- ADP-399
- Non-peptide
- AdipoRon
- (–)-Arctigenin
- Arctiin
- Gramine
- Matairesinol
- Peptide
- Antagonists
- Peptide
- ADP-400
- Peptide
AdipoR2
Main article: Adiponectin receptor 2
- Agonists
- Peptide
- Adiponectin
- ADP-355
- ADP-399
- Non-peptide
- AdipoRon
- Deoxyschizandrin
- Parthenolide
- Syringing
- Taxifoliol
- Peptide
- Antagonists
- Peptide
- ADP-400
- Peptide
Angiotensin receptor
Main article: Angiotensin receptor
Bradykinin receptor
Main article: Bradykinin receptor
- Agonists
- Bradykinin
- Kallidin
- Antagonists
- FR-173657
- Icatibant
- LF22-0542
Cholecystokinin receptor
Main article: Cholecystokinin receptor
CCKA
Main article: Cholecystokinin A receptor
- Agonists
- Cholecystokinin
- Antagonists
- Amiglumide
- Asperlicin
- Devazepide
- Dexloxiglumide
- Lintitript
- Lorglumide
- Loxiglumide
- Pranazepide
- Proglumide
- Tarazepide
- Tomoglumide
CCKB
Main article: Cholecystokinin B receptor
- Agonists
- Cholecystokinin
- CCK-4
- Gastrin
- Pentagastrin (CCK-5)
- Antagonists
- Ceclazepide
- CI-988 (PD-134308)
- Itriglumide
- L-365,360
- Netazepide
- Proglumide
- Spiroglumide
Unsorted
- Antagonists
- Nastorazepide
Corticotropin-releasing hormone receptor
Main article: Corticotropin-releasing hormone receptor
CRF1
Main article: Corticotropin-releasing hormone receptor 1
- Agonists
- Cortagine
- Corticorelin
- Corticotropin-releasing hormone
- Sauvagine
- Stressin I
- Urocortin
- Antagonists
- Antalarmin
- Astressin-B
- CP-154,526
- Emicerfont
- Hypericin
- LWH-234
- NBI-27914
- NBI-74788
- Pexacerfont
- R-121919
- TS-041
- Verucerfont
CRF2
Main article: Corticotropin-releasing hormone receptor 2
- Agonists
- Corticorelin
- Corticotropin-releasing hormone
- Sauvagine
- Urocortin
- Antagonists
- Astressin-B
Cytokine receptor
Main article: Cytokine receptor
Endothelin receptor
Main article: Endothelin receptor
- Agonists
- Endothelin 1
- Endothelin 2
- Endothelin 3
- IRL-1620
- Sarafotoxin
- Antagonists
- A-192621
- Ambrisentan
- Aprocitentan
- Atrasentan
- Avosentan
- Bosentan
- BQ-123
- BQ-788
- Clazosentan
- Darusentan
- Edonentan
- Enrasentan
- Fandosentan
- Feloprentan
- Macitentan
- Nebentan
- Sitaxentan
- Sparsentan
- Tezosentan
- Zibotentan
Galanin receptor
Main article: Galanin receptor
GAL1
Main article: Galanin receptor 1
- Agonists
- Galanin
- Galanin (1-15)
- Galanin-like peptide
- Galmic
- Galnon
- NAX 810-2
- Antagonists
- C7
- Dithiepine-1,1,4,4-tetroxide
- Galantide (M15)
- M32
- M35
- M40
- SCH-202596
GAL2
Main article: Galanin receptor 2
- Agonists
- Galanin
- Galanin (1-15)
- Galanin (2-11)
- Galanin-like peptide
- Galmic
- Galnon
- J18
- NAX 810-2
- Antagonists
- C7
- Galantide (M15)
- M32
- M35
- M40
- M871
GAL3
Main article: Galanin receptor 3
- Agonists
- Galanin
- Galanin (1-15)
- Galmic
- Galnon
- Antagonists
- C7
- Galantide (M15)
- GalR3ant
- HT-2157
- M32
- M35
- M40
- SNAP-37889
- SNAP-398299
Growth hormone secretagogue receptor
Main article: Growth hormone secretagogue receptor
Growth hormone receptor
Main article: Growth hormone receptor
Growth-hormone-releasing hormone receptor
Main article: Growth-hormone-releasing hormone receptor
Glucagon-like peptide receptor
GLP-1
Main article: Glucagon-like peptide-1 receptor
- Agonists
- Albiglutide
- Beinaglutide
- Dulaglutide
- Efpeglenatide
- Exenatide
- GLP-1
- Langlenatide
- Liraglutide
- Lixisenatide
- Oxyntomodulin
- Pegapamodutide
- Semaglutide
- Taspoglutide
GLP-2
Main article: Glucagon-like peptide-2 receptor
- Agonists
- Apraglutide
- Elsiglutide
- Glepaglutide
- GLP-2
- Teduglutide
Others
- Propeptides
- Preproglucagon
- Proglucagon
Glucagon receptor
Main article: Glucagon receptor
- Agonists
- Dasiglucagon
- Glucagon
- Oxyntomodulin
- Antagonists
- Adomeglivant
- L-168,049
- LGD-6972
- Propeptides
- Preproglucagon
- Proglucagon
Gonadotropin-releasing hormone receptor
Main article: Gonadotropin-releasing hormone receptor
Gonadotropin receptor
Main article: Gonadotropin receptor
Growth factor receptor
Main article: Growth factor receptor
Insulin receptor
Main article: Insulin receptor
- Agonists
- Chaetochromin (4548-G05)
- Insulin-like growth factor 1
- Insulin-like growth factor 2
- Insulin
- Insulin aspart
- Insulin degludec
- Insulin detemir
- Insulin glargine
- Insulin glulisine
- Insulin lispro
- Mecasermin
- Mecasermin rinfabate
- Antagonists
- BMS-754807
- S661
- S961
- Kinase inhibitors
- Linsitinib
- Antibodies
- Xentuzumab (against IGF-1 and IGF-2)
KiSS1-derived peptide receptor
Main article: KiSS1-derived peptide receptor
- Agonists
- Kisspeptin (kisspeptin-54, metastin)
- Kisspeptin-10
- KISS1-305
- MVT-602 (RVT-602, TAK-448)
- TAK-683
- Antagonists
- Kisspeptin-234
Leptin receptor
Main article: Leptin receptor
- Agonists
- Leptin
- Metreleptin
Melanin-concentrating hormone receptor
Main article: Melanin-concentrating hormone receptor
MCH1
Main article: Melanin-concentrating hormone receptor 1
- Agonists
- Melanin-concentrating hormone
- Antagonists
- ATC-0065
- ATC-0175
- GW-803430
- NGD-4715
- SNAP-7941
- SNAP-94847
MCH2
Main article: Melanin-concentrating hormone receptor 2
- Agonists
- Melanin-concentrating hormone
Melanocortin receptor
Main article: Melanocortin receptor
Neuropeptide FF receptor
Main article: Neuropeptide FF receptor
- Agonists
- Neuropeptide AF
- Neuropeptide FF
- Neuropeptide SF (RFRP-1)
- Neuropeptide VF (RFRP-3)
- Antagonists
- BIBP-3226
- RF9
Neuropeptide S receptor
Main article: Neuropeptide S receptor
- Agonists
- Neuropeptide S
- Antagonists
- ML-154
- SHA-68
Neuropeptide Y receptor
Main article: Neuropeptide Y receptor
Y1
Main article: Neuropeptide Y receptor Y1
- Agonists
- Neuropeptide Y
- Peptide YY
- Antagonists
- BIBO-3304
- BIBP-3226
- BVD-10
- GR-231118
- PD-160170
Y2
Main article: Neuropeptide Y receptor Y2
- Agonists
- 2-Thiouridine 5'-triphosphate
- Neuropeptide Y
- Neuropeptide Y (13-36)
- Peptide YY
- Peptide YY (3-36)
- Antagonists
- BIIE-0246
- JNJ-5207787
- SF-11
Y4
- Agonists
- GR-231118
- Neuropeptide Y
- Pancreatic polypeptide
- Peptide YY
- Antagonists
- UR-AK49
Y5
Main article: Neuropeptide Y receptor Y5
- Agonists
- BWX-46
- Neuropeptide Y
- Peptide YY
- Antagonists
- CGP-71683
- FMS-586
- L-152,804
- Lu AA-33810
- MK-0557
- NTNCB
- Velneperit (S-2367)
Neurotensin receptor
Main article: Neurotensin receptor
NTS1
Main article: Neurotensin receptor 1
- Agonists
- Neurotensin
- Neuromedin N
- Antagonists
- Meclinertant
- SR-142948
NTS2
Main article: Neurotensin receptor 2
- Agonists
- Neurotensin
- Antagonists
- Levocabastine
- SR-142948
- Levocabastine
Opioid receptor
Main article: Opioid receptor
Orexin receptor
Main article: Orexin receptor
Oxytocin receptor
Main article: Oxytocin receptor
Prolactin receptor
Main article: Prolactin receptor
Parathyroid hormone receptor
Main article: Parathyroid hormone receptor
- Agonists
- Abaloparatide
- Parathyroid hormone
- Parathyroid hormone-related protein (PTHrP)
- Semparatide
- Teriparatide
Relaxin receptor
Main article: Relaxin receptor
- Agonists
- Insulin-like factor 3
- Relaxin (1, 2, 3)
- Serelaxin
Somatostatin receptor
Main article: Somatostatin receptor
Tachykinin receptor
Main article: Tachykinin receptor
Thyrotropin-releasing hormone receptor
Main article: Thyrotropin-releasing hormone receptor
- Agonists
- Azetirelin
- JTP-2942
- Montirelin
- Orotirelin
- Posatirelin
- Protirelin
- Rovatirelin
- RX-77368 (thymoliberin)
- Taltirelin
- TRH (TRF)
Thyrotropin receptor
Main article: Thyrotropin receptor
- Agonists
- Thyrotropin alfa
- TSH (thyrotropin)
Vasopressin receptor
Main article: Vasopressin receptor
Vasoactive intestinal peptide receptor and Pituitary adenylate cyclase-activating peptide
Main article: Vasopressin receptor
VIPR1
Main article: VIPR1
- Agonists
- Peptide
- Bay 55-9837
- LBT-3393
- PACAP
- VIP
- Peptide
VIPR2
Main article: VIPR2
- Agonists
- Peptide
- LBT-3627
- PACAP
- VIP
- Peptide
PAC1
Main article: ADCYAP1R1
- Agonists
- PACAP
- PACAP (1-27)
- PACAP (1-38)
- Antagonists
- PACAP (6-38)
Unsorted
- PHI
- PHM
- PHV
Others
- Endogenous
- Adrenomedullin
- Apelin
- Asprosin
- Bombesin
- Calcitonin
- Carnosine
- CART
- CLIP
- DSIP
- Enteroglucagon
- Formyl peptide
- GALP
- GIP
- GRP
- Integrin ligands
- collagens
- fibrinogen
- fibronectin
- laminins
- ICAM-1
- ICAM-2
- osteopontin
- VCAM-1
- vitronectin
- Kininogens
- Motilin
- Natriuretic peptides
- ANP
- BNP
- CNP
- urodilatin
- Nesfatin-1
- Neuromedin B
- Neuromedin N
- Neuromedin S
- Neuromedin U
- Obestatin
- Osteocalcin
- Resistin
- Secretin
- Thymopoietin
- Thymosins
- Thymulin
- Urotensin-II
- VGF
- Exogenous
- Lifitegrast (LFA-1 antagonist)
References
This article was imported from Wikipedia and is available under the Creative Commons Attribution-ShareAlike 4.0 License. Content has been adapted to SurfDoc format. Original contributors can be found on the article history page.
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