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Etazocine

Chemical compound

10286-45-0 ((−)-form (HCl)) or 5,7-diethyl-2-hydroxy-2-methyl-6,7-benzomorphan GPA-208 ((−)-form); GPA-2087 ((−)-form); NIH-8178 ((−)-form); FDA-0487 ((−)-form) | elimination_half-life =

Etazocine (NIH-7856) is an opioid analgesic of the benzomorphan family which was never marketed. It acts as a partial agonist of the opioid receptors, with mixed agonist and antagonist effects. In animal studies, it was shown to induce analgesia, dependency, and respiratory depression, with overall effects similar to those of morphine, but with substantially reduced potency in comparison.

References

(1969). "Bulletin, problems of drug dependence". National Academies.
(December 1971). "The respiratory effects of a potent analgesic (GPA 2087) in man". British Journal of Anaesthesia.
National Research Council (U.S.). Committee on Problems of Drug Dependence. (1970). "Report of the annual scientific meeting". National Research Council.

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hydroxyarenes benzomorphans opioids

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